產(chǎn)品名稱 Rolofylline metabolite M1-trans - Compound 3
產(chǎn)品貨號 Axon 1851 CAS [160943-06-6] MF C20H28N4O3MW 372.46 Purity: 99% Soluble in DMSO Description Active metabolite of Rolofylline (Axon 1603), a potent and selective adenosine A1 receptor antagonist References Certificates Categories Extra info W Radziszewski et al. A single supratherapeutic dose of rolofylline does not prolong the QTcF interval in healthy volunteers. Am. J. Ther. 2010, 17(1), 8-16. ? M Stroh et al. The Effects of Multiple Doses of Rolofylline on the Single-Dose Pharmacokinetics of Midazolam in Healthy Subjects. Am. J. Ther. 2010, 17(1), 53-60.? Certificate of Analysis Material Safety Data Sheet CNS A1 A18 Adenosine A1 antagonist Chemical name 8-(Hexahydro-7-hydroxy-2,5-methanopentalen-3a(1H)-yl)-3,9-dihydro-1,3-dipropyl-1H-Purine-2,6-dione, trans Parent CAS No. [160943-06-6] Order Size Unit Price Stock 2 mg €105.00 In Stock
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Rolofylline metabolite M1-trans - Compound 3

Based on 15 reference(s) in Google Scholar 8 10 15

Axon 1851

CAS [160943-06-6]

MF C20H28N4O3
MW 372.46

  • Purity: 99%
  • Soluble in DMSO

Rolofylline metabolite M1-trans

Description

Active metabolite of Rolofylline (Axon 1603), a potent and selective adenosine A1 receptor antagonist

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