產(chǎn)品名稱 SGC2085
產(chǎn)品貨號 Axon 2625 CAS [1821908-49-9] MF C19H24N2O2.HClMW 348.87 Purity: 100% Soluble in water and DMSO Description Potent and selective Coactivator Associated Arginine Methyltransferase 1 (CARM1 or PRMT4) inhibitor (IC50 value 50 nM and >100-fold selectivity over other PRMTs). Unfortunately, no cellular activity was observed for SGC2085 when tested up to 10 μM due to due to poor cell permeability (in HEK293 cells). KEYWORDS:?SGC2085 | supplier | CARM1 inhibitor | SGC-2085 | CAS [1821908-49-9] | [1821908-48-8] | Arginine | PRMT4 | Coactivator Associated Arginine Methyltransferase 1 | oncology | Wnt | β-Catenin
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
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產(chǎn)品品牌 axonmedchem
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SGC2085

Based on 1 publications in PubMed 9 10 1

Axon 2625

CAS [1821908-49-9]

MF C19H24N2O2.HCl
MW 348.87

  • Purity: 100%
  • Soluble in water and DMSO

SGC2085

Description

Potent and selective Coactivator Associated Arginine Methyltransferase 1 (CARM1 or PRMT4) inhibitor (IC50 value 50 nM and >100-fold selectivity over other PRMTs). Unfortunately, no cellular activity was observed for SGC2085 when tested up to 10 μM due to due to poor cell permeability (in HEK293 cells).

KEYWORDS:?SGC2085 | supplier | CARM1 inhibitor | SGC-2085 | CAS [1821908-49-9] | [1821908-48-8] | Arginine | PRMT4 | Coactivator Associated Arginine Methyltransferase 1 | oncology | Wnt | β-Catenin

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