| 產(chǎn)品名稱 | AM 251 |
| 產(chǎn)品貨號(hào) | Axon 1218 CAS [183232-66-8] MF C22H21Cl2IN4OMW 555.24 Purity: 99% Soluble in DMSO and Ethanol Description Cannabinoids CB1 antagonist, structurally very close to SR 141716A (rimonabant). AM251: Ki 7.5 nM for CB1 receptor vs SR 141716A ( Ki value of 11.5 nM). However AM251 is about two-fold more selective for the CB1 receptor when compared to SR 141716A References Certificates Categories Extra info R Lan et al. Structure-activity relationships of pyrazole derivatives as cannabinoid receptor antagonists. J. Med. Chem. 1999, 42 769-776. Certificate of Analysis Material Safety Data Sheet Cardiovascular CNS Diabetes & Metabolism Pain & Inflammation CB1 A13 CB1 antagonist Chemical name 1-(2,4-Dichloro-phenyl)-5-(4-iodo-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide Parent CAS No. [183232-66-8] Order Size Unit Price Stock 10 mg €95.00 In Stock |
| 產(chǎn)品價(jià)格 | 現(xiàn)貨詢價(jià)，電話：010-67529703 |
| 產(chǎn)品規(guī)格 | |
| 產(chǎn)品品牌 | axonmedchem |
| 產(chǎn)品概述 | |
| 產(chǎn)品詳情 |
AM 251Axon 1218 CAS [183232-66-8] MF C22H21Cl2IN4O
Description
Cannabinoids CB1 antagonist, structurally very close to SR 141716A (rimonabant). AM251: Ki 7.5 nM for CB1 receptor vs SR 141716A ( Ki value of 11.5 nM). However AM251 is about two-fold more selective for the CB1 receptor when compared to SR 141716A
CB1 antagonist
Chemical name1-(2,4-Dichloro-phenyl)-5-(4-iodo-phenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide Parent CAS No.[183232-66-8] |
| 產(chǎn)品資料 |
