產(chǎn)品名稱 Lapatinib ditosylate - GW 572016
產(chǎn)品貨號(hào) Axon 1395 CAS [388082-77-7] MF C29H26ClFN4O4S.2C7H8O3SMW 925.46 Purity: 99% Soluble in DMSO Description An ATP-competitive epidermal growth factor receptor (EGFR) and HER2/neu (ErbB-2) dual tyrosine kinase inhibitor References Certificates Categories Extra info HA Burris. Dual kinase inhibition in the treatment of breast cancer: initial experience with the EGFR/ErbB-2 inhibitor lapatinib. Oncologist 2004, 9 Suppl 3: 10–5. ? MH Nelson, CR Dolder. Lapatinib: a novel dual tyrosine kinase inhibitor with activity in solid tumors. Ann Pharmacother 2006, 40(2), 261–9. Certificate of Analysis Material Safety Data Sheet Angiogenesis Cell Signaling & Oncology EGFR ErbB2-HER2 JAK-STAT RTK class I; EC 2.7.10.1 EGFR and ErbB-2/HER2 tyrosine kinase inhibitor Chemical name N-[3-chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[(2-methylsulfonylethylamino)methyl]-2-furyl] quinazolin-4-amine ditosylate Parent CAS No. [231277-92-2] Order Size Unit Price Stock 10 mg €95.00 In Stock
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Lapatinib ditosylate - GW 572016

Based on 16 reference(s) in Google Scholar 9 10 16

Axon 1395

CAS [388082-77-7]

MF C29H26ClFN4O4S.2C7H8O3S
MW 925.46

  • Purity: 99%
  • Soluble in DMSO

Lapatinib ditosylate

Description

An ATP-competitive epidermal growth factor receptor (EGFR) and HER2/neu (ErbB-2) dual tyrosine kinase inhibitor
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