產(chǎn)品名稱 TCS1102
產(chǎn)品貨號 Axon 2744 CAS [916141-36-1] MF C27H26N4O2SMW 470.59 Purity: 98% Optical purity: Optically pure Soluble in DMSO Description TCS1102 is a potent and selective dual orexin receptor antagonist (Ki values of 3 and 0.2 nM for hOX1R and hOX2R, respectively). Moreover, TCS1102 demonstrated in vivo central activity when dosed peripherally in a pharmacodynamic model of orexin activity. KEYWORDS: TCS1102 | supplier | OX1/2 antagonist | TCS 1102 | TCS-1102 | DORA-1 | DORA1 | DORA 1 | CAS [916141-36-1] | Orexin | Orexin (OX) | Antagonist | Receptors
產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
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產(chǎn)品品牌 axonmedchem
產(chǎn)品概述
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TCS1102

Based on 11 reference(s) in Google Scholar 8 10 11

Axon 2744

CAS [916141-36-1]

MF C27H26N4O2S
MW 470.59

  • Purity: 98%
  • Optical purity: Optically pure
  • Soluble in DMSO

TCS1102

Description

TCS1102 is a potent and selective dual orexin receptor antagonist (Ki values of 3 and 0.2 nM for hOX1R and hOX2R, respectively). Moreover, TCS1102 demonstrated in vivo central activity when dosed peripherally in a pharmacodynamic model of orexin activity.

KEYWORDS: TCS1102 | supplier | OX1/2 antagonist | TCS 1102 | TCS-1102 | DORA-1 | DORA1 | DORA 1 | CAS [916141-36-1] | Orexin | Orexin (OX) | Antagonist | Receptors

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