Selective BRD7 and BRD9 inhibitor (Kd values are 99 and 909 nM, respectively). Exhibits selectivity for BRD7/9 over a panel of 48 bromodomains (at 10 μM). Inhibits interactions with histones H3.3 and H4 at low micromolar concentrations. Decreases the level of IL-6 secreted from LPS-stimulated THP-1 cells. Negative control ent-LP 99 (Cat.No. 5497) also available. Purity 98%. MW (observed): 516.05