產(chǎn)品名稱 CID 16020046 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 4959/25
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 25 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameCID 16020046
    DescriptionSelective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21 μM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase, μ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice. Purity 99%. MW (observed): 425.44
    Size25 mg
    Concentrationn/a
    Applicationsn/a
    Other Names4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid
    Gene, Accession, CAS #CAS: 834903-43-4
    Catalog #4959/25
    Price
    Order / More InfoCID 16020046 from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 25989290, 28552522, 28779174, 28800762
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