產(chǎn)品名稱 GNE 2861 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 6490/5
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 5 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameGNE 2861
    DescriptionInhibitor of group II p21 activated kinases (PAK; IC50 values are 7.5, 126 and 36 nM for PAK4, PAK5 and PAK6, respectively). Displays selectivity for group II PAK over a panel of 222 kinases. Inhibits tumor cell proliferation, migration and invasion in two breast cancer cell lines. Also sensitizes tamoxifen-resistant breast cancer cell lines to tamoxifen (Cat. No. 6342) via PAK4-dependent regulation of estrogen receptor α (ERα) target gene expression. Purity 98%. MW (observed): 406.48
    Size5 mg
    Concentrationn/a
    Applicationsn/a
    Other Names1-[2-[1-(2-Amino-4-pyrimidinyl)-2-[(2-methoxyethyl)amino]-1H-benzimidazol-6-yl]ethynyl]cyclohexanol
    Gene, Accession, CAS #CAS: 1394121-05-1
    Catalog #6490/5
    Price
    Order / More InfoGNE 2861 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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