產(chǎn)品名稱 CHMFL-FLT3-122 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 5800/50
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 50 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameCHMFL-FLT3-122
    DescriptionPotent and selective FLT3 inhibitor (IC50 = 40 nM). Exhibits >10-fold and 170-fold selectivity for FLT3 over BTK kinase and c-KIT kinase, respectively in vitro. Induces apoptosis by arresting cell cycle in G0/G1 phase in vitro. Suppresses tumor growth in an AML xenograft model. Modestly orally bioavailable. MW (observed): 471.55.
    Size50 mg
    Concentrationn/a
    Applicationsn/a
    Other Names1-[(3R)-3-[4-Amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]-1-piperidinyl]-2-(dimethylamino)-ethanone
    Gene, Accession, CAS #CAS: 1839150-56-9
    Catalog #5800/50
    Price
    Order / More InfoCHMFL-FLT3-122 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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