產(chǎn)品名稱 RQ 00203078 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 5388/10
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameRQ 00203078
    DescriptionPotent TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively). Exhibits >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1. Reduces HSC3 and HSC4 oral squamous carcinoma cell migration and invasion in vitro. Also attenuates icilin -induced wet dog shakes in rats. Orally active. Purity 98%. MW (observed): 554.85
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other Names4-[[[3-Chloro-5-(trifluoromethyl)-2-pyridinyl][[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]benzoic acid
    Gene, Accession, CAS #CAS: 1254205-52-1
    Catalog #5388/10
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    Order / More InfoRQ 00203078 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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