產(chǎn)品名稱 GSK-2126458 from BIOVISION, INC.
    產(chǎn)品貨號 1961-5
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 5 mg
    產(chǎn)品品牌 BIOVISION, INC.
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameGSK-2126458
    DescriptionCell-permeable. A highly potent, pan phosphoinositide 3-kinase (PI 3-K) family kinase inhibitor with biochemical Ki's of 0.019 nM (PI 3-Kα), 0.13 nM (PI 3-Kβ), 0.024 nM (PI 3-Kδ), 0.06 nM (PI 3-Kγ), 0.18 nM (mTORC1), and 0.3 nM (mTORC2). In vivo, GSK2126458 displays anti-tumor activity in both pharmacodynamic and tumor growth efficacy models. MW: 505.5. Purity ≥98% by HPLC
    Size5 mg
    Concentrationn/a
    Applicationsn/a
    Other Names2,4-Difluoro-N-{2-(methyloxy)-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl}benzenesulfonamide
    Gene, Accession, CAS #CAS: 1086062-66-9
    Catalog #1961-5
    Price
    Order / More InfoGSK-2126458 from BIOVISION, INC.
    Product Specific Referencesn/a
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