A highly selective, potent small molecule inhibitor of RORγ; inhibits RORγ transactivation in cell lines at 0.1-10 μM; inhibits IL-17A and IL-22 secretion from cultured human Th17 cells (IC50 = 3.2 nM)
Size
25 mg
Concentration
n/a
Applications
n/a
Other Names
GSK-2981278 RAR ROR-g RORg IL17A IL22 chinese hamster ovary interleukin