產(chǎn)品名稱 PD 135158 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 2608/10
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
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    Product NamePD 135158
    DescriptionPotent and selective, nonpeptide CCK2 receptor antagonist (IC50 values are 2.8 and 1232 nM for CCK2 and CCK1 respectively) that displays negligible affinity at GABAA, benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT3 receptors (IC50 > 10 μM). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats. Purity 98%. MW (observed): 616.76
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other Names4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid. CAM 1028
    Gene, Accession, CAS #CAS: 130285-87-9
    Catalog #2608/10
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    Order / More InfoPD 135158 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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