產(chǎn)品名稱 PND-1186 from BIOVISION, INC.
    產(chǎn)品貨號(hào) 2823-5
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 5 mg
    產(chǎn)品品牌 BIOVISION, INC.
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NamePND-1186
    DescriptionPND-1186 is a potent FAK (Focal adhesion kinase) inhibitor (IC50 = 1.5 nM) with potential antineoplastic activity. PND-1186 inhibits FAK, blocks fibronectin-stimulated FAK autophosphorylation of Tyr397, and may prevent the integrin-mediated activation of several downstream signal transduction pathways, including ERK, JNK/MAPK and PI3K/Akt. This results in the reduction of the number of cancer stem cells (CSCs) and inhibits tumor cell migration, proliferation and survival. MW: 501.5. Purity ≥98% by HPLC
    Size5 mg
    Concentrationn/a
    Applicationsn/a
    Other Names2-((2-((2-methoxy-4-morpholinophenyl)amino)-5-(trifluoromethyl)pyridin-4-yl)amino)-N-methylbenzamide; VS-4718; SR-2516;PND 1186;PND1186;SR 2516;SR2516
    Gene, Accession, CAS #CAS: 1061353-68-1
    Catalog #2823-5
    Price
    Order / More InfoPND-1186 from BIOVISION, INC.
    Product Specific Referencesn/a
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