產(chǎn)品名稱 (+/-)-AMG 487 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 4487/10
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
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    Product Name(+/-)-AMG 487
    DescriptionAntagonist of CXCR3; inhibits binding of 125I-IP-10 and 125I-ITAC to CXCR3 (IC50 values are 8.0 and 8.2 nM respectively). Inhibits CXCR3-mediated cell migration by the chemokines IP-10, ITAC and MiG in vitro (IC50 values are 8, 15 and 36 nM respectively). Also shown to inhibit lung metastasis in a mouse model of metastatic breast cancer. This product is racemic. . Purity 98%. MW (observed): 603.59
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other NamesN-1-[(3-4(-Ethoxyphenyl)-3,4-dihydro-4-oxopyrido[2,3-d]pyrimidin-2-yl]ethyl]-N-(3-pyridinylmethyl)-4-(trifluoromethoxy)benzeneacetamide
    Gene, Accession, CAS #CAS: 947536-03-0
    Catalog #4487/10
    Price
    Order / More Info(+/-)-AMG 487 from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 28986561, 30359318
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