產(chǎn)品名稱 PF 03814735 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 4821/50
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 50 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
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    Product NamePF 03814735
    DescriptionATP-competitive inhibitor of Aurora kinases A and B (IC50 values are 0.8 and 5 nM for recombinant Aurora B and Aurora A, respectively). Inhibits phosphorylation of Aurora B, histone H3 and Aurora A in cultured MDA-MB-231 cells (IC50 values are approximately 20, 50 and 150 nM respectively). Shown to block cytokinesis; inhibits cellular proliferation in several human tumor cell lines, including HCT-116, HL-60, A549 and H125, and in human xenograft mouse models. Orally available. Purity 98%. MW (observed): 474.48
    Size50 mg
    Concentrationn/a
    Applicationsn/a
    Other NamesN-[2-[(1S,4R)-6-[[4-(Cyclobutylamino)-5-(trifluoromethyl)-2-pyrimidinyl]amino]-1,2,3,4-tetrahydronaphthalen-1,4-imin-9-yl]-2-oxoethyl]-acetamide
    Gene, Accession, CAS #CAS: 942487-16-3
    Catalog #4821/50
    Price
    Order / More InfoPF 03814735 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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