產(chǎn)品名稱 (+/-)-NBI 74330 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 4528/10
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product Name(+/-)-NBI 74330
    DescriptionPotent and selective CXCR3 antagonist; potently inhibits 125I-CXCL10 binding to CXCR3 (pKi = 8.13). Inhibits calcium mobilization in response to CXCL11 and CXCL10 in RBL cells. Exhibits no significant effect on chemotaxis induced by CXCR4 or CCR7. Displays a five-fold greater affinity for CXCR3 than (±)-AMG 487. This product is racemic. . Purity 98%. MW (observed): 605.58
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other NamesN-1-[(3-4(-Ethoxyphenyl)-3,4-dihydro-4-oxopyrido[2,3-d]pyrimidin-2-yl]ethyl]-4-fluoro-N-(3-pyridinylmethyl)-3-(trifluoromethyl)benzeneacetamide
    Gene, Accession, CAS #CAS: 473722-68-8
    Catalog #4528/10
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    Order / More Info(+/-)-NBI 74330 from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 30076959
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