產(chǎn)品名稱 ERK5-IN-1 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 5393/50
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 50 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameERK5-IN-1
    DescriptionPotent and selective ERK5 inhibitor; inhibits EGFR-induced ERK5 autophosphorylation (EC50 = 90 nM) and ERK5 enzymatic activity (IC50 = 162 nM). Exhibits at least 30-fold selectivity for ERK5 over LRRK2 in a cell based assay. Also selective for ERK5 over a panel of other kinases. Orally bioavailable. Purity 98%. MW (observed): 638.8
    Size50 mg
    Concentrationn/a
    Applicationsn/a
    Other Names11-Cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
    Gene, Accession, CAS #CAS: 1435488-37-1
    Catalog #5393/50
    Price
    Order / More InfoERK5-IN-1 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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