產(chǎn)品名稱 FR 180204 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 3706/10
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameFR 180204
    DescriptionSelective ERK inhibitor (IC50 values are 0.14 and 0.31 μM for ERK2 and ERK1 respectively). Displays 30-fold selectivity for ERK over p38α (IC50 = 10 μM); displays no activity against human recombinant MEK1, MKK4, IKKα, PKCα, Src, Syc and PDGFα at concentrations less than 30 μM. Also inhibits TGFβ-induced AP-1 activation in Mv1Lu cells (IC50 = 3.1 μM). Purity 98%. MW (observed): 327.34
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other Names5-(2-Phenyl-pyrazolo[1,5-a]pyridin-3-yl)-1H-pyrazolo[3,4-c]pyridazin-3-ylamine
    Gene, Accession, CAS #CAS: 865362-74-9
    Catalog #3706/10
    Price
    Order / More InfoFR 180204 from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 22683469, 24086109, 25052197, 25195011, 25425646, 25547114, 25738359, 27659207
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