產(chǎn)品名稱 PF 3644022 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 4279/10
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
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    Product NamePF 3644022
    DescriptionPotent, ATP-competitive inhibitor of mitogen-activated protein kinase (MAPK)-activated protein kinase-2 (MK2) (IC50 = 5.2 nM; Ki = 3 nM). Inhibits tumor necrosis factor α (TNFα) production in U937 monocytic cells and peripheral blood mononuclear cells (PBMCs) (IC50 = 160 nM); exhibits oral efficacy in acute and chronic inflammatory models. Purity 98%. MW (observed): 374.46
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other Names(10R)-9,10,11,12-Tetrahydro-10-methyl-3-(6-methyl-3-pyridinyl)-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one
    Gene, Accession, CAS #CAS: 1276121-88-0
    Catalog #4279/10
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    Order / More InfoPF 3644022 from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 26017782, 28506461
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