產(chǎn)品名稱 BRL 54443 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 1129/10
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameBRL 54443
    DescriptionA potent 5-ht1E/1F receptor agonist (pEC50 values are 8.5 and 8.6 respectively). Displays > 30-fold selectivity over other 5-HT and dopamine receptors (pKi values are 8.7. 8.9, 7.2, 6.9, 7.2, 5.9, 7.0, 6.5, < 6, < 6, 6.3 and 6.2 for human 5-HT1E, 1F, 1A, 1B, 1D, 2A, 2B, 2C, 4, 7, D2 and D3 receptors respectively). Induces 5-HT2A receptor-mediated mouse aortic contraction in vitro (pEC50 = 6.52). Active in vivo. MW (observed): 230.31.
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other Names5-Hydroxy-3-(1-methylpiperidin-4-yl)-1H-indole
    Gene, Accession, CAS #CAS: 57477-39-1
    Catalog #1129/10
    Price
    Order / More InfoBRL 54443 from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 19649285, 21422162
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