產(chǎn)品名稱 INCB 3284 dimesylate from TOCRIS BIOSCIENCE
    產(chǎn)品貨號 4306/10
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 10 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameINCB 3284 dimesylate
    DescriptionPotent, selective hCCR2 antagonist. Exhibits potent antagonism against monocyte chemoattractant molecule binding to hCCR2 and chemotaxis activity (IC50 values are 3.7 and 4.7 nM respectively). Also displays weak hERG activity; inhibits the hERG potassium current (IC50 = 84μM). Orally bioavailable. Purity 98%. MW (observed): 712.76
    Size10 mg
    Concentrationn/a
    Applicationsn/a
    Other NamesN-[2-[[(3R)-1-[trans-4-Hydroxy-4-(6-methoxy-3-pyridinyl)cyclohexyl]-3-pyrrolidinyl]amino]-2-oxoethyl]-3-(trifluoromethyl)-benzamide dimethanesulfonate
    Gene, Accession, CAS #CAS: 887401-93-6
    Catalog #4306/10
    Price
    Order / More InfoINCB 3284 dimesylate from TOCRIS BIOSCIENCE
    Product Specific ReferencesPubMed: 24904083, 25012628, 27216982
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