產(chǎn)品名稱 AZ 6102 from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 5775/50
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 50 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameAZ 6102
    DescriptionPotent TNKS2 and TNKS1 inhibitor (IC50 values are 1 and 3 nM, respectively). Exhibits >100-fold selectivity for TNKS1/2 over PARP-1, PARP-2 and PARP-6. Inhibits Wnt signaling in DLD-1 cells (IC50 = 5 nM). Exhibits moderate oral bioavailability. Purity 98%. MW (observed): 428.53
    Size50 mg
    Concentrationn/a
    Applicationsn/a
    Other Namesrel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one
    Gene, Accession, CAS #CAS: 1645286-75-4
    Catalog #5775/50
    Price
    Order / More InfoAZ 6102 from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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