產(chǎn)品名稱 Lonafarnib from TOCRIS BIOSCIENCE
    產(chǎn)品貨號(hào) 6265/50
    產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
    產(chǎn)品規(guī)格 50 mg
    產(chǎn)品品牌 TOCRIS BIOSCIENCE
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameLonafarnib
    DescriptionPotent farnesyl transferase inhibitor (IC50 = 1.9 nM). Inhibits farnesylation of RAS. Also inhibits Pgp transport (IC50 < 3 μM) and increases potency and anticancer activity when used in conjunction with cytotoxic Pgp substrates. Inhibits neovascularization by affecting cell motility. Orally bioavailable. Purity 98%. MW (observed): 638.82
    Size50 mg
    Concentrationn/a
    Applicationsn/a
    Other Names4-[2-[4-[(11R)-3,10-Dibromo-8-chloro-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-yl]-1-piperidinyl]-2-oxoethyl]-1-piperidinecarboxamide
    Gene, Accession, CAS #CAS: 193275-84-2
    Catalog #6265/50
    Price
    Order / More InfoLonafarnib from TOCRIS BIOSCIENCE
    Product Specific Referencesn/a
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