A benzoic acid derivative that inhibits OAT1, OAT3, and OAT6 with Ki values of 6.3, 9.0, and 8.4 μM, respectively, as well as OAT2 with an IC50 value of 0.67 μM; enhances the renal excretion of urate while reducing the elimination of many medications; acts as an agonist of TRPV2 (EC50 = 31.9 μM)