產(chǎn)品名稱 RVX-208 from CAYMAN CHEMICAL COMPANY
    產(chǎn)品貨號 16424-5
    產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
    產(chǎn)品規(guī)格 5 mg
    產(chǎn)品品牌 CAYMAN CHEMICAL COMPANY
    產(chǎn)品概述
    產(chǎn)品詳情
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    Product NameRVX-208
    DescriptionA selective antagonist of BET bromodomains, binding with 10-100-fold higher affinity for BD2 (IC50 = 0.04-0.28 μM) over BD1 (IC50 = 1.8-3.1 μM), which causes selective release of BET proteins from chromatin; increases the expression of ApoA1 and reduces atherosclerosis in hyperlipidemic ApoE-deficient mice
    Size5 mg
    Concentrationn/a
    Applicationsn/a
    Other Namesepigenetics atherosclerosis proteins bindings chromatins research BD1 BD2 BDs 1 2 ones twos BD-1 BD-2 RVXs RVX208 208 bromodomains selective antagonists BETs cells apolipoproteins ApoA1 A1 mice mouse monkeys humans hyperlipidemic ApoE deficient deficiency deficiencies 1246400-89-4 1431550-07-0 RVX 000222 biochemicals
    Gene, Accession, CAS #CAS: 1044870-39-4
    Catalog #16424-5
    Price
    Order / More InfoRVX-208 from CAYMAN CHEMICAL COMPANY
    Product Specific Referencesn/a
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